XRPD Method Development & Validation

Custom XRPD method development for polymorph quantification and pharmaceutical QC

Overview

At DANNALAB we can detect and quantify polymorphic impurities down to a limit of as low as parts of % wt. For finished dosage forms, in some cases, we are able to validate detection limit (LOD) down to 0.17% and quantification limit (LOQ) as low as 0.5% wt from total.

Why is this important? XRPD is a method specifically for the identification of polymorphs. The investigation of polymorphs (chemically identical substances in different crystallographic forms) is a key step in drug product development. Since polymorphic forms differ in their solid-state structure, they can have different aqueous solubilities and dissolution rates.

Presence of minor traces of patented polymorphic impurity may have significant legal implications as well.

Related Application Note

XRPD Quantification of Polymorph Impurities →

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